SCHEMBL10259495

SCHEMBL10259495

COc1ccc(CNC(=O)N2[C@H]3CN(Cc4ccco4)C(=O)C(CCC(=O)O)N3C(=O)CN2C)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 10/20 0.43
ALDH1A1 P00352 2/20 0.39
APOBEC3A P31941 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CLPP Q16740 2/20 0.38
CACNA1G O43497 1/20 0.38
CACNA1H O95180 1/20 0.38
CACNA1I Q9P0X4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL749624 1.00 CYP3A4 (0.43) CYP3A4ALDH1A1APOBEC3AAPOBEC3GMEN1
SCHEMBL746731 0.93 CYP3A4 (0.43) CYP3A4ALDH1A1APOBEC3AAPOBEC3GMEN1
SCHEMBL749613 0.93 CYP3A4 (0.44) CYP3A4ALDH1A1APOBEC3AAPOBEC3GMEN1
SCHEMBL747387 0.93 CLPP (0.43) CYP3A4ALDH1A1POLBCLPP
SCHEMBL749671 0.91 PKM (0.42) CYP3A4ALDH1A1APOBEC3AAPOBEC3GMEN1
SCHEMBL745982 0.91 CYP3A4 (0.38) CYP3A4LMNASMN1; SMN2CLPP
SCHEMBL749607 0.91 CLPP (0.46) CYP3A4ALDH1A1APOBEC3AAPOBEC3GSMN1; SMN2
SCHEMBL750691 0.91 CYP3A4 (0.52) CYP3A4CLPP
SCHEMBL749577 0.90 CYP3A4 (0.46) CYP3A4MEN1KMT2ACLPPCACNA1G
SCHEMBL745988 0.90 MEN1 (0.49) CYP3A4MEN1KMT2ACLPPCACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101751-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-01-24 US disclosed
US-8101751-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-01-24 US disclosed