SCHEMBL10262153

SCHEMBL10262153

COc1ccc(C2(c3ccc(OC)cc3)C=Cc3c4c(c5cc(N(C)C)c(-c6ccc(N7CCOCC7)cc6)cc5c3O2)-c2ccccc2C42CC(C)(C)CC(C)(C)C2)cc1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 4/20 0.34
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
AKT1 P31749 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13868646 0.95 PRKDC (0.36) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL10267979 0.94 PRKDC (0.33) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL13868628 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL10267980 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL13868685 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL10292860 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL13868630 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL10262395 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL10262462 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1
SCHEMBL15449577 0.93 PRKDC (0.34) PRKDCPIK3CDPIK3CAAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8691120-B2 Chromene compound TOKUYAMA CORPORATION (JP) 2014-04-08 US disclosed
US-8691120-B2 Chromene compound TOKUYAMA CORPORATION (JP) 2014-04-08 US disclosed
US-20120170098-A1 CHROMENE COMPOUND TOKUYAMA CORPORATION (JP) 2012-07-05 US disclosed
US-20120170098-A1 CHROMENE COMPOUND TOKUYAMA CORPORATION (JP) 2012-07-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120170098-A1 CHROMENE COMPOUND CRY2, CRY1, SUN2 PRKDC 2990/4885PIK3CD 2854/4885PIK3CA 2002/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.