SCHEMBL10264407

SCHEMBL10264407

O=C1CCc2cc(C(=O)N3CCNCC3)[nH]c21

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 9/20 0.49
HRH3 Q9Y5N1 1/20 0.49
SIGMAR1 Q99720 1/20 0.44
HPGD P15428 1/20 0.38
HSP90AA1 P07900 1/20 0.38
PARP1 P09874 2/20 0.38
RHEB Q15382 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13562313 0.85 HRH4 (0.59) HRH4HRH3
SCHEMBL10263146 0.77 HRH4 (0.64) HRH4HRH3
SCHEMBL1006834 0.76 ALOX15 (0.48) HPGD
SCHEMBL10263385 0.75 HRH4 (0.74) HRH4HRH3SIGMAR1HPGDHSP90AA1
SCHEMBL10263701 0.75 HRH4 (0.69) HRH4HRH3SIGMAR1HPGDHSP90AA1
SCHEMBL10264424 0.71 HRH4 (0.47) HRH4HRH3SIGMAR1HSP90AA1RHEB
SCHEMBL10264652 0.70 HRH4 (0.49) HRH4HRH3SIGMAR1HSP90AA1RHEB
SCHEMBL10263610 0.70 HRH4 (0.49) HRH4HRH3SIGMAR1HSP90AA1RHEB
SCHEMBL13562341 0.69 HRH4 (0.47) HRH4HRH3SIGMAR1HSP90AA1RHEB
SCHEMBL13562353 0.69 HRH4 (0.47) HRH4HRH3SIGMAR1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460794-A1 PHARMACEUTICAL COMPOSITION CONTAINING FUSED HETERO-RING DERIVATIVE Shionogi & Co., Ltd. (JP) 2012-06-06 EP disclosed