SCHEMBL10265129

SCHEMBL10265129

COC(=O)c1sc(C(C)(C)C)cc1NC1CCN(C)C(=O)C1

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 17/20 0.45
MAPK14 Q16539 8/20 0.45
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL325364 0.83 NR1I2 (0.38) RAF1
SCHEMBL10264745 0.82 RAF1 (0.49) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10206941 0.79 RAF1 (0.50) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL12514492 0.79 ALDH1A1 (0.47) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10264797 0.78 RAF1 (0.48) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL14670273 0.78 RAF1 (0.51) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10268700 0.77 RAF1 (0.47) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL12520070 0.77 RAF1 (0.50) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL9965153 0.75 RAF1 (0.48) RAF1MAPK14MAPK13MAPK12MAPK11
SCHEMBL10265010 0.73 RAF1 (0.50) RAF1MAPK14MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006055-A2 COMPOUNDS AND METHODS FOR THE TREATMENT OR PREVENTION OF FLAVIVIRUS INFECTIONS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-01-12 WO disclosed