SCHEMBL1027003

SCHEMBL1027003

CC(C)(C)C(c1cc(N(COCC[Si](C)(C)C)COCC[Si](C)(C)C)n2ncc(-c3cnc4ccccc4c3)c2n1)N(C(=O)O)C1CCOCC1

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.32
JAK1 P23458 1/20 0.32
JAK3 P52333 1/20 0.32
AVPR1B P47901 1/20 0.32
TTK P33981 2/20 0.31
PIK3CA P42336 1/20 0.31
GPR119 Q8TDV5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1074594 0.87 HSP90AA1 (0.32) HSP90AA1JAK1JAK3AVPR1B
SCHEMBL1023161 0.83 HSP90AA1 (0.34) HSP90AA1JAK1JAK3AVPR1BTTK
SCHEMBL593155 0.82
SCHEMBL1027004 0.81 HSP90AA1 (0.32) HSP90AA1JAK1JAK3AVPR1BPIK3CA
SCHEMBL6890894 0.80 JAK1 (0.36) HSP90AA1JAK1JAK3AVPR1BTTK
SCHEMBL1073468 0.77 JAK1 (0.37) HSP90AA1JAK1JAK3PIK3CA
SCHEMBL1082183 0.77 JAK1 (0.34) HSP90AA1JAK1JAK3AVPR1BTTK
SCHEMBL2679521 0.76 SMO (0.37) HSP90AA1AVPR1BPIK3CA
SCHEMBL584040 0.76 ATR (0.41) PIK3CA
SCHEMBL7879162 0.76 RAB9A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002887-A1 FUSED TRICYCLIC COMPOUNDS AS NOVEL mTOR INHIBITORS SCHERING CORPORATION (US) 2011-01-06 WO disclosed