SCHEMBL7879162

SCHEMBL7879162

Cc1cc(N(COCC[Si](C)(C)C)COCC[Si](C)(C)C)n2ncc(-c3cnc4ccccc4c3)c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 11/20 0.39
MAPT P10636 11/20 0.39
NPC1 O15118 9/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
KMT2A Q03164 7/20 0.38
KDM4E B2RXH2 6/20 0.38
MEN1 O00255 6/20 0.38
ALDH1A1 P00352 5/20 0.38
HSD17B10 Q99714 4/20 0.38
MAPK1 P28482 3/20 0.38
TP53 P04637 3/20 0.38
HPGD P15428 3/20 0.38
TSHR P16473 2/20 0.38
ALOX15 P16050 1/20 0.38
GFER P55789 1/20 0.38
CRHR1 P34998 4/20 0.36
STAT1 P42224 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
NR2F2 P24468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31339 0.90 KDM4E (0.33) RAB9AMAPTNPC1SMN1; SMN2KMT2A
SCHEMBL1083466 0.88 AKR1C3 (0.32)
SCHEMBL583888 0.88 RAB9A (0.32) RAB9AMAPTNPC1L3MBTL1KMT2A
SCHEMBL12461451 0.85 MAPT (0.41) RAB9AMAPTNPC1SMN1; SMN2L3MBTL1
SCHEMBL584040 0.85 ATR (0.41) RAB9AMAPTNPC1SMN1; SMN2KMT2A
SCHEMBL10238601 0.84 PDE10A (0.33) RAB9AMAPTNPC1SMN1; SMN2KDM4E
SCHEMBL584192 0.83 HSP90AA1 (0.38) RAB9AMAPTNPC1SMN1; SMN2KMT2A
SCHEMBL10238603 0.83 PDE10A (0.32)
SCHEMBL617633 0.83
SCHEMBL10280192 0.82 CHRNB1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118207-A1 PYRAZOLO [1, 5-A] PYRIMIDINE DERIVATIVES AS MTOR INHIBITORS SCHERING CORPORATION (US) 2010-10-14 WO disclosed