1,2,3,4-Tetrahydroisoquinoline

1,2,3,4-Tetrahydroisoquinoline

SCHEMBL1027366

O=C(NO)C1NCc2ccccc21.c1ccc2c(c1)CCNC2

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.50
CD44 P16070 1/20 0.50
MAOB P27338 1/20 0.50
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HDAC4 P56524 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
HTR2C P28335 2/20 0.39
OPRM1 P35372 5/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36
F2 P00734 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32689446 0.82 TSHR (0.67) TSHRNPSR1HDAC4HDAC7HDAC5
SCHEMBL5160890 0.82 TSHR (0.67) TSHRNPSR1HDAC4HDAC7HDAC5
SCHEMBL24113114 0.74 TSHR (0.44) TSHRNPSR1HDAC4HDAC7HDAC5
SCHEMBL4163569 0.73 TSHR (0.44) TSHRNPSR1OPRM1F2
1,2,3,4-Tetrahydroisoquinoline SCHEMBL6010101 0.73 PNMT (0.79) PNMTCD44MAOBHTR2C
SCHEMBL4164018 0.72 SMYD3 (0.43) TSHRNPSR1HDAC4HDAC7HDAC5
1,2,3,4-Tetrahydroisoquinoline SCHEMBL4779021 0.71 PNMT (0.76) PNMTCD44MAOBHTR2C
SCHEMBL27632988 0.71 TSHR (0.50) TSHRNPSR1
1,2,3,4-Tetrahydroisoquinoline SCHEMBL29360217 0.71 PNMT (1.00) PNMTCD44MAOBHTR2C
1,2,3,4-Tetrahydroisoquinoline SCHEMBL28236302 0.71 PNMT (1.00) PNMTCD44MAOBHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274283-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2011-01-19 EP disclosed
WO-2009112550-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2009-09-17 WO disclosed