SCHEMBL10273685

SCHEMBL10273685

Cc1ccncc1-c1ccc(NS(=O)(=O)C2CC2)cc1O

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 11/20 0.64
PRMT6 Q96LA8 1/20 0.44
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
JAK1 P23458 2/20 0.42
ABL1 P00519 1/20 0.41
CKS1B P61024 1/20 0.40
SKP2 Q13309 1/20 0.40
BRPF1 P55201 1/20 0.39
MAP4K1 Q92918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL527428 0.90 CYP17A1 (0.67) CYP17A1PRMT6PTGS1PTGS2JAK1
SCHEMBL526869 0.83 CYP17A1 (0.70) CYP17A1PTGS1PTGS2
SCHEMBL527268 0.82 PRMT6 (0.58) CYP17A1PRMT6PTGS1PTGS2ABL1
SCHEMBL15746951 0.79 CYP17A1 (1.00) CYP17A1PRMT6
SCHEMBL526391 0.72 CYP17A1 (0.78) CYP17A1PTGS1PTGS2
SCHEMBL527762 0.71 CYP17A1 (0.48) CYP17A1ABL1
SCHEMBL526628 0.70 CYP17A1 (0.59) CYP17A1PTGS1PTGS2
SCHEMBL527415 0.70 CYP17A1 (0.59) CYP17A1PTGS1PTGS2
SCHEMBL18112987 0.70 BRPF1 (0.45) CYP17A1BRPF1
SCHEMBL526755 0.69 CYP17A1 (0.76) CYP17A1PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012015723-A1 SULFONAMIDE COMPOUNDS USEFUL AS CYP17 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-02 WO disclosed