SCHEMBL10276687

SCHEMBL10276687

Cc1cc(B2OC(C)(C)C(C)(C)O2)ccc1-c1ncnn1COCC[Si](C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
F2RL1 P55085 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.32
DGAT1 O75907 4/20 0.32
LPL P06858 3/20 0.31
LIPG Q9Y5X9 3/20 0.31
HIF1A Q16665 1/20 0.31
SNCA P37840 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1442542 0.92 DGAT1 (0.33) F2RL1IRAK4DGAT1LPLLIPG
SCHEMBL1440509 0.90 DGAT1 (0.38) F2RL1IRAK4DGAT1LPLLIPG
SCHEMBL10276614 0.86 LPL (0.40) F2RL1DGAT1LPLLIPGSNCA
SCHEMBL16283835 0.81 PRMT5 (0.32) DGAT1CA1CA2CA9
SCHEMBL1440712 0.80 F2RL1 (0.36) F2RL1DGAT1LPLLIPG
SCHEMBL1440522 0.80 F2RL1 (0.33) F2RL1DGAT1
SCHEMBL1441281 0.79 DGAT1 (0.46) F2RL1DGAT1
SCHEMBL1442282 0.78 DGAT1 (0.32) IRAK4DGAT1LPLLIPGHIF1A
SCHEMBL10276963 0.78 F2RL1 (0.32) F2RL1
SCHEMBL1444504 0.76 F2RL1 (0.37) F2RL1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8865726-B2 Substituted pyrazolo[1,5-a]pyrimidine compounds as mTOR inhibitors ARRAY BIOPHARMA INC. (US) 2014-10-21 US disclosed
US-20120178715-A1 SUBSTITUTED PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS ARRAY BIOPHARMA INC. (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178715-A1 SUBSTITUTED PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS MTOR, RICTOR, EIF4EBP1 F2RL1 3780/4885IRAK4 2469/4885DGAT1 4722/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.