SCHEMBL10278912

SCHEMBL10278912

C=C(C)CCNc1cnc(N)cn1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
HCAR3 P49019 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037308 0.77 KDM4E (0.47) JAK2TYK2ALDH1A1
SCHEMBL2645239 0.72 HCAR3 (0.49) HCAR3ALDH1A1
SCHEMBL2644724 0.68 ALOX5AP (0.33) HCAR3
SCHEMBL5040443 0.67 L3MBTL1 (0.50) ALDH1A1
SCHEMBL16680902 0.66 MEN1 (0.36)
SCHEMBL14390105 0.65
SCHEMBL20714407 0.63 MAPT (0.52) ALDH1A1
SCHEMBL4253816 0.63
SCHEMBL5044824 0.62 HCAR3 (0.43) JAK2JAK3HCAR3
SCHEMBL16388495 0.62 IKBKE (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020008-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE F. HOFFMANN-LA ROCHE AG (CH) 2012-02-16 WO disclosed