SCHEMBL10282917

SCHEMBL10282917

BCc1cc(CN(CCOC)C(=O)OC(C)(C)C)cc(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
ROCK2 O75116 2/20 0.35
HDAC1 Q13547 4/20 0.34
HDAC3 O15379 2/20 0.34
HDAC2 Q92769 2/20 0.34
NCOR2 Q9Y618 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
SSTR4 P31391 1/20 0.33
MLYCD O95822 1/20 0.33
TACR1 P25103 1/20 0.32
HDAC6 Q9UBN7 1/20 0.31
BACE1 P56817 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL89599 0.89 GRIN2D (0.40) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL89601 0.88 GRIN2D (0.39) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL8262797 0.86 GRIN2D (0.38) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL8263905 0.84 HDAC1 (0.38) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL90346 0.82 ALDH1A1 (0.45) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL1800114 0.74 CYP4F2 (0.42) ROCK2HDAC1HDAC3HDAC2NCOR2
SCHEMBL13166745 0.74 HDAC1 (0.45) HDAC1HDAC3HDAC2NCOR2L3MBTL1
SCHEMBL1800104 0.73 HDAC1 (0.44) HDAC1HDAC3HDAC2NCOR2SSTR4
SCHEMBL3567836 0.72 RIPK1 (0.46) ROCK2HDAC1HDAC3HDAC2NCOR2
SCHEMBL28987476 0.72 PPARG (0.47) HDAC1HDAC3HDAC2NCOR2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2420491-A1 3 , 5-substitued piperidine compounds as renin inhibitors Novartis AG (CH) 2012-02-22 EP disclosed