SCHEMBL10288142

SCHEMBL10288142

Nc1c(N2CCOCC2)sc(-c2nnn[nH]2)c1Cc1ccc2ccccc2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.36
TPH1 P17752 1/20 0.32
PRKDC P78527 1/20 0.32
CETP P11597 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
GAA P10253 2/20 0.31
MAPT P10636 2/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
CYP2D6 P10635 1/20 0.31
NFKB1 P19838 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
PIK3CA P42336 2/20 0.31
HTR6 P50406 1/20 0.31
PTPN1 P18031 1/20 0.31
AKT1 P31749 1/20 0.31
KMT2A Q03164 1/20 0.31
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627366 0.86 PIK3CA (0.40) PIK3CAPIK3CDPIK3CGPIK3CB
SCHEMBL10298513 0.86 PDE10A (0.34) PDE10APRKDCCETP
SCHEMBL626480 0.80 NPC1 (0.37) PDE10APRKDCCETPALDH1A1HPGD
SCHEMBL10288131 0.75 HSD17B10 (0.42) PDE10ATPH1PRKDCKDM4EALDH1A1
SCHEMBL10298533 0.69 KDM4E (0.32) KDM4EALDH1A1MAPTPIK3CA
SCHEMBL952623 0.68 MPO (0.37) PDE10ACETPCYP2D6NFKB1TAAR1
SCHEMBL10288613 0.65 TRPV1 (0.37) KDM4EALDH1A1GAAMAPTHPGD
SCHEMBL16850491 0.65 PDE10A (0.41) PDE10ACETPALDH1A1PIK3CAPIK3CD
SCHEMBL623933 0.64 PIK3CA (0.52) TPH1KDM4EALDH1A1MAPTHPGD
SCHEMBL10298521 0.64 AKR1C3 (0.38) PDE10ATPH1PRKDCKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021696-A1 HETEROARYLS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-16 WO disclosed