SCHEMBL952623

SCHEMBL952623

Nc1cccc(-c2nnn[nH]2)c1Cc1ccc2ccccc2c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.37
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
BACE1 P56817 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
PDE10A Q9Y233 3/20 0.33
CETP P11597 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2A6 P11509 1/20 0.33
EGFR P00533 1/20 0.32
FLT1 P17948 1/20 0.32
CHEK2 O96017 1/20 0.32
NQO1 P15559 1/20 0.32
ALOX5 P09917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL951950 0.79 TP53 (0.38) MPOCYP2D6CHEK2
SCHEMBL949313 0.76 MPO (0.42) MPOCYP2D6NFKB1TAAR1BACE1
SCHEMBL1247974 0.72 CYP2D6 (0.46) MPOCYP2D6NFKB1TAAR1BACE1
SCHEMBL3277728 0.72 ALDH1A1 (0.52)
SCHEMBL30940314 0.72 ALDH1A1 (0.52)
SCHEMBL6775919 0.71 DHFR (0.42) NFKB1ADORA2AADORA1CYP1A2ALOX5
Hydrochloric Acid SCHEMBL27778340 0.70 ALDH1A1 (0.50)
SCHEMBL11146024 0.69 ALDH1A1 (0.38)
SCHEMBL9423544 0.68 ALDH1A1 (0.35) CYP1A2
SCHEMBL3745750 0.67 HCAR2 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2454243-A2 TETRAZOLE DERIVATIVES Merck Serono SA (CH) 2012-05-23 EP disclosed
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed