SCHEMBL10288591

SCHEMBL10288591

CC(c1ccc2cc(F)ccc2c1)c1c(C=O)sc(N2CCOCC2)c1C#N

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.36
PIK3CG P48736 4/20 0.36
PIK3R1 P27986 4/20 0.36
PIK3CD O00329 3/20 0.36
PIK3CB P42338 3/20 0.36
MTOR P42345 2/20 0.36
HPGD P15428 2/20 0.35
MAPK1 P28482 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CTSL P07711 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KCNQ2 O43526 1/20 0.33
CYP3A4 P08684 1/20 0.33
KDM4E B2RXH2 4/20 0.33
ALDH1A1 P00352 3/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 2/20 0.33
GPR6 P46095 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10288574 0.91 HPGD (0.38) PIK3CAPIK3R1MTORHPGDMAPK1
SCHEMBL10308557 0.87 HPGD (0.36) PIK3CAPIK3CGPIK3R1PIK3CDPIK3CB
SCHEMBL10288604 0.84 PIK3CA (0.48) PIK3CAPIK3CGPIK3R1PIK3CDPIK3CB
SCHEMBL10288409 0.81 ALDH1A1 (0.37) PIK3CAPIK3CGPIK3R1PIK3CDPIK3CB
SCHEMBL10288572 0.79 KDM4E (0.38) PIK3CAPIK3CGPIK3R1PIK3CDPIK3CB
SCHEMBL10288594 0.78 ALDH1A1 (0.36) PIK3CAPIK3CGPIK3R1PIK3CDPIK3CB
SCHEMBL10288607 0.77 SLC6A2 (0.36) PIK3CAPIK3R1HPGDMAPK1NPSR1
SCHEMBL10308588 0.77 HPGD (0.38) PIK3CAHPGDMAPK1NPSR1SMN1; SMN2
SCHEMBL10288191 0.76 PIK3CA (0.35) PIK3CAPIK3R1HPGDMAPK1NPSR1
SCHEMBL625724 0.75 PIK3CA (0.49) PIK3CAPIK3R1PIK3CDPIK3CBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021696-A1 HETEROARYLS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-16 WO disclosed