SCHEMBL10288607

SCHEMBL10288607

COCC(c1ccc2ccccc2c1)c1c(C=O)sc(N2CCOCC2)c1C#N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
KCNH2 Q12809 1/20 0.36
ALDH1A1 P00352 2/20 0.36
PIK3CA P42336 4/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
PIK3R1 P27986 2/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
APP P05067 1/20 0.33
USP9X Q93008 1/20 0.32
CDK1 P06493 1/20 0.32
CDK4 P11802 1/20 0.32
CCNB1 P14635 1/20 0.32
CCNA2 P20248 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10288594 0.89 ALDH1A1 (0.36) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL10298720 0.86 PIK3CA (0.46) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL10288574 0.86 HPGD (0.38) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL10288409 0.84 ALDH1A1 (0.37) ALDH1A1PIK3CAHPGDKDM4EHSD17B10
SCHEMBL10288191 0.83 PIK3CA (0.35) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL10288591 0.77 PIK3CA (0.36) CYP3A4ALDH1A1PIK3CAHPGDKDM4E
SCHEMBL622922 0.76 PIK3CA (0.47) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL10298686 0.75 HPGD (0.36) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL10288569 0.75 PIK3CA (0.46) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL623045 0.74 PIK3CA (0.41) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012021696-A1 HETEROARYLS AND USES THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-16 WO disclosed