SCHEMBL10290993

SCHEMBL10290993

CCC(=O)Nc1cc(C(=O)NC(C)c2ccc(N)nc2)cc(C)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
RAB9A P51151 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ADORA3 P0DMS8 6/20 0.38
ADORA1 P30542 4/20 0.38
P2RX3 P56373 4/20 0.38
P2RX2 Q9UBL9 4/20 0.38
ALDH1A1 P00352 1/20 0.37
HPGDS O60760 2/20 0.37
ADORA2A P29274 3/20 0.36
ADORA2B P29275 1/20 0.36
MAPK1 P28482 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
NR1I2 O75469 1/20 0.35
CYP2C9 P11712 1/20 0.35
KLKB1 P03952 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4550460 0.84 NPC1 (0.42) NPC1POLBRAB9ATDP1ADORA3
SCHEMBL2717586 0.83 ACACB (0.40) NPC1POLBRAB9ATDP1P2RX3
SCHEMBL2716878 0.83 MAPK1 (0.38) NPC1POLBRAB9ATDP1ADORA3
SCHEMBL2715471 0.83 NR1I2 (0.38) NPC1POLBRAB9ATDP1ADORA3
SCHEMBL2713996 0.82 EPHX2 (0.40) P2RX3P2RX2NR1I2CYP2C9
SCHEMBL2715036 0.81 NR1I2 (0.39) P2RX3P2RX2ALDH1A1NR1I2CYP2C9
SCHEMBL2716275 0.81 EPHX2 (0.39) P2RX3P2RX2NR1I2CYP2C9ACACB
SCHEMBL2713943 0.81 SCN9A (0.37) P2RX3P2RX2ALDH1A1NR1I2CYP2C9
SCHEMBL2714167 0.80 SCN9A (0.36) P2RX3P2RX2ALDH1A1NR1I2CYP2C9
SCHEMBL2713828 0.79 LMNA (0.45) NPC1RAB9AP2RX3P2RX2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed