SCHEMBL4550460

SCHEMBL4550460

CCC(=O)Nc1cc(C(=O)NC(C)c2ccc(O)cc2)cc(C)n1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
POLB P06746 1/20 0.42
RAB9A P51151 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
ADORA3 P0DMS8 8/20 0.41
ADORA1 P30542 5/20 0.41
ALDH1A1 P00352 3/20 0.40
ADORA2A P29274 4/20 0.39
ADORA2B P29275 3/20 0.39
LMNA P02545 2/20 0.39
PDE2A O00408 1/20 0.39
TSHR P16473 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2718591 0.84 PDE2A (0.52) PDE2A
SCHEMBL10290993 0.84 NPC1 (0.39) NPC1POLBRAB9ATDP1ADORA3
SCHEMBL2713828 0.83 LMNA (0.45) NPC1RAB9AALDH1A1LMNAPDE2A
SCHEMBL2716055 0.80 GPR139 (0.47) NPC1POLBRAB9ATDP1LMNA
SCHEMBL2716053 0.80 GPR139 (0.47) NPC1POLBRAB9ATDP1LMNA
SCHEMBL2716878 0.79 MAPK1 (0.38) NPC1POLBRAB9ATDP1ADORA3
SCHEMBL2717586 0.79 ACACB (0.40) NPC1POLBRAB9ATDP1ALDH1A1
SCHEMBL2715471 0.79 NR1I2 (0.38) NPC1POLBRAB9ATDP1ADORA3
SCHEMBL18266123 0.79 NPC1 (0.41) NPC1POLBRAB9ATDP1ADORA3
SCHEMBL18266582 0.79 ALDH1A1 (0.52) ADORA3ADORA1ALDH1A1ADORA2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed