SCHEMBL1030734

SCHEMBL1030734

COc1ccc(-c2c(C)cn(Cc3ccc(F)cc3)c2C(=O)NCCN(C)C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.45
CNR2 P34972 3/20 0.45
FAAH O00519 2/20 0.45
CYP2D6 P10635 2/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
HSD17B10 Q99714 1/20 0.40
LMNA P02545 3/20 0.40
TP53 P04637 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
MAPT P10636 3/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ABHD6 Q9BV23 1/20 0.39
RAD52 P43351 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1031481 0.84 THRB (0.53) CNR1CNR2FAAHGLALMNA
SCHEMBL1031690 0.82 HPGD (0.46) CNR1CNR2FAAHALDH1A1HPGD
SCHEMBL2637247 0.82 CHRM1 (0.47) CNR1CNR2FAAHKDM4EALDH1A1
SCHEMBL1032507 0.80 PPARG (0.49) CNR1CNR2FAAHKDM4EALDH1A1
SCHEMBL1032474 0.80 NPC1 (0.44) ALDH1A1HPGDLMNATP53MEN1
SCHEMBL1028497 0.79 PRKAA2 (0.44) KDM4EALDH1A1LMNAMAPT
SCHEMBL1031104 0.79 CNR1 (0.43) CNR1CNR2FAAHKDM4EALDH1A1
SCHEMBL1030364 0.79 MCHR1 (0.47) CNR1CNR2CYP2D6KDM4EALDH1A1
SCHEMBL1032118 0.79 POLB (0.40) CNR1KDM4EALDH1A1HPGDLMNA
SCHEMBL1029726 0.77 PTGS2 (0.52) MAPTKMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed