SCHEMBL10312195

SCHEMBL10312195

Cc1cc(Nc2nc(/C=C/c3cccc(F)c3)nc(NCc3ccncc3)n2)n[nH]1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PAK4 O96013 4/20 0.48
PLK4 O00444 3/20 0.48
NTRK1 P04629 14/20 0.46
NTRK3 Q16288 2/20 0.45
NTRK2 Q16620 2/20 0.45
AURKA O14965 1/20 0.45
DAPK3 O43293 1/20 0.45
JAK2 O60674 1/20 0.45
ABL1 P00519 1/20 0.45
LCK P06239 1/20 0.45
FYN P06241 1/20 0.45
CSF1R P07333 1/20 0.45
RET P07949 1/20 0.45
IGF1R P08069 1/20 0.45
PDGFRB P09619 1/20 0.45
FGFR1 P11362 1/20 0.45
FLT1 P17948 1/20 0.45
LTK P29376 1/20 0.45
KDR P35968 1/20 0.45
FLT3 P36888 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10312189 0.90 PAK4 (0.51) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312205 0.89 KCNH3 (0.40) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL16556867 0.89 PAK4 (0.45) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312107 0.89 PAK4 (0.49) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312224 0.88 NTRK1 (0.50) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312211 0.85 IGF1R (0.50) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312218 0.84 NTRK1 (0.44) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312221 0.81 HRH4 (0.48) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312187 0.81 AURKA (0.42) PAK4PLK4NTRK1NTRK3NTRK2
SCHEMBL10312198 0.79 IGF1R (0.42) PAK4PLK4IGF1RFGFR1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440055-B1 STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS CALIFORNIA CAPITAL EQUITY LLC (US) 2015-03-11 EP disclosed
US-20120178758-A1 STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS CALIFORNIA CAPITAL EQUITY, LLC (US) 2012-07-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120178758-A1 STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS STK25, STK35, SGK2 PAK4 254/4885PLK4 287/4885NTRK1 482/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.