SCHEMBL1032074

SCHEMBL1032074

CCn1cc(C)c(-c2ccc(Cl)cc2)c1C(=O)NCC(C)c1ccc(Cl)cc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 3/20 0.39
MDM2 Q00987 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
P2RX7 Q99572 4/20 0.37
MAPT P10636 2/20 0.36
EP300 Q09472 2/20 0.36
OPRM1 P35372 1/20 0.35
BCL2 P10415 5/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BCL2L1 Q07817 4/20 0.35
MCL1 Q07820 4/20 0.35
BCL2A1 Q16548 4/20 0.35
BAK1 Q16611 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1748908 0.80 GCGR (0.43) BCL2
SCHEMBL2637730 0.77 GRIA2 (0.45) RAB9ANPC1TP53MDM2MAPT
SCHEMBL1031754 0.75 KDM4E (0.52) RAB9ANPC1TDP1MAPTMEN1
SCHEMBL1031856 0.74 BCL2 (0.35) TP53MDM2MAPTEP300BCL2
SCHEMBL1031707 0.73 POLB (0.46) TP53MDM2MAPTBCL2MEN1
SCHEMBL1031726 0.73 KDM4E (0.49) RAB9ANPC1MAPTMEN1KMT2A
SCHEMBL1030036 0.73 HSP90AA1 (0.38) TDP1MAPTKMT2A
SCHEMBL1030744 0.72 POLB (0.47) TP53MAPTBCL2MEN1KMT2A
SCHEMBL1031910 0.70 NPC1 (0.59) RAB9ANPC1MEN1KMT2A
SCHEMBL1031266 0.70 CCR1 (0.44) TDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed