SCHEMBL10322010

SCHEMBL10322010

CN(c1ccc(-n2ccc3cc(N(CC(=O)O)S(=O)(=O)c4cc(Cl)cc(Cl)c4)ccc32)nn1)C1CCOCC1.CN(c1ccc(I)nn1)C1CCOCC1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 3/20 0.32
NFE2L2 Q16236 3/20 0.32
ALDH1A1 P00352 2/20 0.31
USP2 O75604 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3301557 0.96 ALDH1A1 (0.34) KEAP1NFE2L2ALDH1A1USP2TSHR
SCHEMBL13390727 0.87 TSHR (0.32) ALDH1A1USP2TSHR
SCHEMBL4432779 0.86 KEAP1 (0.35) KEAP1NFE2L2ALDH1A1
SCHEMBL3298686 0.85 KEAP1 (0.35) KEAP1NFE2L2ALDH1A1USP2TSHR
SCHEMBL10318086 0.83 KEAP1 (0.36) KEAP1NFE2L2ALDH1A1
SCHEMBL4430841 0.81 KEAP1 (0.39) KEAP1NFE2L2ALDH1A1USP2TSHR
SCHEMBL13409227 0.81 PTGDR2 (0.31)
SCHEMBL3298220 0.81 ALDH1A1 (0.34) KEAP1NFE2L2ALDH1A1USP2TSHR
SCHEMBL3300839 0.81 KEAP1 (0.35) KEAP1NFE2L2ALDH1A1USP2TSHR
SCHEMBL3298351 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121600-B1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INT (DE) 2012-07-18 EP disclosed