SCHEMBL1032776

SCHEMBL1032776

Cc1cn(Cc2ccc(C(F)(F)F)cc2)c(C(=O)Nc2ccc(C(C)(C)C)cc2)c1-c1ccco1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
MEN1 O00255 2/20 0.45
KDM4E B2RXH2 2/20 0.45
HPGD P15428 1/20 0.45
TRPV1 Q8NER1 1/20 0.45
POLB P06746 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
LMNA P02545 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
HIF1A Q16665 3/20 0.42
EPAS1 Q99814 3/20 0.42
NR3C1 P04150 2/20 0.41
MAPT P10636 2/20 0.41
SCD5 Q86SK9 1/20 0.40
RAB9A P51151 2/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1032310 0.83 ADORA2A (0.42) KMT2ACYP1A2CYP2C9CYP2C19KDM4E
SCHEMBL1029856 0.81 HTT (0.46) KMT2ACYP1A2CYP2C9CYP2C19MEN1
SCHEMBL1030837 0.81 NPC1 (0.44) KMT2AMEN1KDM4EHPGDPOLB
SCHEMBL1031730 0.80 CNR1 (0.45) KMT2ACYP2C9CYP2C19MEN1KDM4E
SCHEMBL1031988 0.79 CNR1 (0.44) KMT2ACYP2C9CYP2C19MEN1KDM4E
SCHEMBL1032145 0.79 EPHX2 (0.45)
SCHEMBL1030813 0.77 TSHR (0.46) KMT2ACYP2C9CYP2C19MEN1POLB
SCHEMBL1031836 0.77 MEN1 (0.43) KMT2ACYP2C9MEN1POLBLMNA
SCHEMBL1031640 0.76 ALDH1A1 (0.52) KMT2ACYP1A2CYP2C9CYP2C19MEN1
SCHEMBL1031499 0.76 SMN1; SMN2 (0.41) KMT2ACYP2C19KDM4EHPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed