SCHEMBL1031640

SCHEMBL1031640

COc1ccc(CCNC(=O)c2c(-c3ccco3)c(C)cn2Cc2ccc(C(F)(F)F)cc2)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.52
MAPT P10636 4/20 0.52
HTT P42858 3/20 0.52
LMNA P02545 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
KDM4E B2RXH2 3/20 0.49
POLB P06746 3/20 0.49
KMT2A Q03164 3/20 0.49
USP2 O75604 2/20 0.49
TP53 P04637 2/20 0.49
PKM P14618 2/20 0.49
ALOX15 P16050 2/20 0.49
MAPK1 P28482 2/20 0.49
HSD17B10 Q99714 2/20 0.49
MEN1 O00255 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
THRB P10828 1/20 0.49
HPGD P15428 1/20 0.49
APEX1 P27695 1/20 0.49
CASP1 P29466 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1030837 0.88 NPC1 (0.44) ALDH1A1MAPTHTTLMNASMN1; SMN2
SCHEMBL1029856 0.82 HTT (0.46) ALDH1A1MAPTHTTLMNASMN1; SMN2
SCHEMBL1032145 0.80 EPHX2 (0.45) HTTNPSR1
SCHEMBL1032310 0.80 ADORA2A (0.42) ALDH1A1HTTLMNASMN1; SMN2KDM4E
SCHEMBL1028135 0.78 ALDH1A1 (0.53) ALDH1A1MAPTLMNAKDM4EPOLB
SCHEMBL1031836 0.77 MEN1 (0.43) HTTLMNASMN1; SMN2POLBKMT2A
SCHEMBL1032776 0.76 KMT2A (0.45) ALDH1A1MAPTLMNAKDM4EPOLB
SCHEMBL1030586 0.76 ALDH1A1 (0.41) ALDH1A1MAPTHTTKDM4EPOLB
SCHEMBL1030443 0.76 RAB9A (0.46) ALDH1A1MAPTLMNASMN1; SMN2KDM4E
SCHEMBL1031019 0.76 PLAAT3 (0.42) ALDH1A1HTTSMN1; SMN2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035375-B1 1,3-DISUBSTITUTED 4-METHYL-1H-PYRROLE-2-CARBOXAMIDES AND THEIR USE FOR THE MANUFACTURE OF MEDICAMENTS GRUENENTHAL GMBH (DE) 2011-01-19 EP claimed