SCHEMBL10328445

SCHEMBL10328445

CCOc1ccc(CC2=CC([C@@H]3O[C@H](SC)[C@@H](O)[C@H](O)[C@H]3O)CC=C2Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SLC5A1 P13866 16/20 0.51
SLC5A2 P31639 15/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10292573 1.00 SLC5A1 (0.51) SLC5A1SLC5A2
SCHEMBL12965051 0.85 SLC5A2 (0.50) SLC5A1SLC5A2
SCHEMBL882697 0.82 SLC5A2 (0.37) SLC5A1SLC5A2
SCHEMBL12323556 0.82 SLC5A2 (0.37) SLC5A1SLC5A2
SCHEMBL13964967 0.75 SLC5A1 (0.37) SLC5A1SLC5A2
SCHEMBL12956970 0.74 SLC5A2 (0.39) SLC5A1SLC5A2
SCHEMBL12797197 0.74 SLC5A2 (0.39) SLC5A1SLC5A2
SCHEMBL14215765 0.74 SLC5A2 (0.35) SLC5A1SLC5A2
SCHEMBL13057263 0.74 SLC5A2 (0.41) SLC5A1SLC5A2
SCHEMBL14215830 0.73 SLC5A2 (0.35) SLC5A1SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8217156-B2 Solid forms of (2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(methylthio)tetrahydro-2H-pyran-3,4,5-triol and methods of their use LEXICON PHARMACEUTICALS, INC. (US) 2012-07-10 US disclosed
US-20110218159-A1 METHODS OF USING INHIBITORS OF SODIUM-GLUCOSE COTRANSPORTERS 1 AND 2 LEXICON PHARMACEUTICALS, INC. 2011-09-08 US disclosed
EP-2332947-A1 Solid forms of (2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(methylthio)tetrahydro-2H-pyran-3,4,5-triol and methods of their use Lexicon Pharmaceuticals, Inc. (US) 2011-06-15 EP disclosed
WO-2010009197-A1 SOLID FORMS OF (2S,3R,4R,5S,6R)-2-(4-CHLORO-3-(4-ETHOXYBENZYL)PHENYL)-6-(METHYLTHIO)TETRAHYDRO-2H-PYRAN-3,4,5-TRIOL AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS, INC. (US) 2010-01-21 WO disclosed
US-20100016422-A1 SOLID FORMS OF (2S,3R,4R,5S,6R)-2-(4-CHLORO-3-(4-ETHOXYBENZYL)PHENYL)-6-(METHYLTHIO)TETRAHYDRO-2H-PYRAN-3,4,5-TRIOL AND METHODS OF THEIR USE OXFORD FINANCE LLC, AS COLLATERAL AGENT 2010-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100016422-A1 SOLID FORMS OF (2S,3R,4R,5S,6R)-2-(4-CHLORO-3-(4-ETHOXYBENZYL)PHENYL)-6-(METHYLTHIO)TETRAHYDRO-2H-PYRAN-3,4,5-TRIOL AND METHODS OF THEIR USE TPMT, PYGL, PNPO SLC5A1 354/4885SLC5A2 233/4885
US-20110218159-A1 METHODS OF USING INHIBITORS OF SODIUM-GLUCOSE COTRANSPORTERS 1 AND 2 SLC5A2, SLC5A1, SLC2A2 SLC5A1 2/4885SLC5A2 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.