SCHEMBL10328478

SCHEMBL10328478

Bc1ccc(S(=O)(=O)Nc2ccc(Cc3ccnc4cc(OC)c(OC)cc34)cc2F)cc1C

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AXL P30530 11/20 0.51
KIT P10721 3/20 0.47
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
PDGFRA P16234 1/20 0.38
KDR P35968 1/20 0.38
MET P08581 1/20 0.38
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10328522 0.89 AXL (0.54) AXLKITABCB1ABCC1KEAP1
SCHEMBL10328519 0.88 AXL (0.51) AXLKITABCB1ABCC1
SCHEMBL10328520 0.87 AXL (0.57) AXLKITABCB1ABCC1
SCHEMBL10328493 0.86 AXL (0.59) AXLKITABCB1ABCC1MET
SCHEMBL10328494 0.86 AXL (0.53) AXLKITABCB1ABCC1KDR
SCHEMBL10328498 0.86 AXL (0.68) AXLKITABCB1ABCC1
SCHEMBL10328487 0.86 AXL (0.57) AXLKITABCB1ABCC1PDGFRA
SCHEMBL10328489 0.84 AXL (0.58) AXLKITPDGFRAKDR
SCHEMBL10328499 0.83 AXL (0.52) AXLMET
SCHEMBL10328491 0.82 AXL (0.55) AXLKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed