SCHEMBL10328487

SCHEMBL10328487

COc1cc2nccc(Cc3ccc(NS(=O)(=O)c4cc(F)cc(F)c4)c(F)c3)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AXL P30530 12/20 0.57
KIT P10721 5/20 0.49
KDR P35968 2/20 0.42
PDGFRA P16234 1/20 0.42
FGFR2 P21802 1/20 0.42
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
FGFR1 P11362 1/20 0.40
FLT1 P17948 1/20 0.40
MET P08581 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10328498 0.91 AXL (0.68) AXLKITABCB1ABCC1
SCHEMBL10328522 0.90 AXL (0.54) AXLKITABCB1ABCC1
SCHEMBL10328520 0.90 AXL (0.57) AXLKITABCB1ABCC1
SCHEMBL10328494 0.87 AXL (0.53) AXLKITKDRABCB1ABCC1
SCHEMBL10328493 0.87 AXL (0.59) AXLKITABCB1ABCC1MET
SCHEMBL10328486 0.86 AXL (0.69) AXLKITKDRFGFR1FLT1
SCHEMBL13667521 0.86 AXL (0.61) AXLKIT
SCHEMBL10328519 0.86 AXL (0.51) AXLKITABCB1ABCC1
SCHEMBL10328478 0.86 AXL (0.51) AXLKITKDRPDGFRAABCB1
SCHEMBL10328489 0.85 AXL (0.58) AXLKITKDRPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed