SCHEMBL10328489

SCHEMBL10328489

COc1cc2nccc(Cc3ccc(NS(=O)(=O)c4cc(C)c(C)cc4OC)c(F)c3)c2cc1OC

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AXL P30530 14/20 0.58
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KIT P10721 3/20 0.43
ALPL P05186 1/20 0.41
PDGFRA P16234 1/20 0.40
KDR P35968 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13667521 0.88 AXL (0.61) AXLKIT
SCHEMBL13667523 0.88 AXL (0.59) AXLKIT
SCHEMBL10328506 0.86 AXL (0.57) AXL
SCHEMBL10328481 0.86 AXL (0.59) AXLKITKDR
SCHEMBL10328503 0.86 AXL (0.59) AXLKIT
SCHEMBL10328498 0.85 AXL (0.68) AXLKIT
SCHEMBL10328487 0.85 AXL (0.57) AXLKITPDGFRAKDR
SCHEMBL10328479 0.85 AXL (0.58) AXLKIT
SCHEMBL10328522 0.84 AXL (0.54) AXLKIT
SCHEMBL10328520 0.84 AXL (0.57) AXLKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed