SCHEMBL10328481

SCHEMBL10328481

COc1cc2nccc(Cc3ccc(NS(=O)(=O)c4ccc(Cl)cc4F)c(F)c3)c2cc1OC

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AXL P30530 10/20 0.59
FLT1 P17948 3/20 0.50
KDR P35968 3/20 0.50
FGFR1 P11362 2/20 0.50
EPHB2 P29323 1/20 0.46
FLT4 P35916 1/20 0.46
SLC40A1 Q9NP59 2/20 0.46
NUDT1 P36639 2/20 0.45
KIT P10721 1/20 0.44
SRC P12931 1/20 0.44
PIK3CA P42336 1/20 0.44
CSF1R P07333 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13667521 0.88 AXL (0.61) AXLKIT
SCHEMBL10328506 0.87 AXL (0.57) AXL
SCHEMBL13667268 0.86 AXL (0.51) AXLFLT1KDRFGFR1KIT
SCHEMBL10328494 0.86 AXL (0.53) AXLFLT1KDRFGFR1KIT
SCHEMBL10328489 0.86 AXL (0.58) AXLKDRKIT
SCHEMBL10328486 0.85 AXL (0.69) AXLFLT1KDRFGFR1KIT
SCHEMBL10328522 0.85 AXL (0.54) AXLKIT
SCHEMBL13667523 0.84 AXL (0.59) AXLSLC40A1KIT
SCHEMBL10328503 0.84 AXL (0.59) AXLKIT
SCHEMBL10328487 0.84 AXL (0.57) AXLFLT1KDRFGFR1KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed