SCHEMBL10328516

SCHEMBL10328516

COc1cc(NS(=O)(=O)c2ccccc2OC(F)(F)F)ccc1Cc1ccnc2cc(OC)c(OC)cc12

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AXL P30530 19/20 0.57
EGFR P00533 2/20 0.56
MET P08581 2/20 0.56
SRC P12931 2/20 0.56
ALPL P05186 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13667478 0.95 AXL (0.57) AXLEGFRMETSRCALPL
SCHEMBL10328526 0.90 AXL (0.58) AXLEGFRMETSRCALPL
SCHEMBL13667283 0.88 AXL (0.48) AXLEGFRMETSRC
SCHEMBL1590945 0.85 AXL (0.78) AXLEGFRMETSRC
SCHEMBL10328530 0.83 AXL (0.73) AXLEGFRMETSRC
SCHEMBL1591743 0.82 AXL (0.79) AXLEGFRMETSRC
SCHEMBL10328505 0.82 AXL (0.73) AXLEGFRMETSRC
SCHEMBL13667556 0.81 AXL (0.70) AXLEGFRMETSRC
SCHEMBL1592214 0.81 AXL (0.78) AXLEGFRMETSRC
SCHEMBL1591652 0.81 AXL (0.79) AXLEGFRMETSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed