SCHEMBL10328526

SCHEMBL10328526

COc1cc2nccc(Cc3ccc(NS(=O)(=O)c4ccccc4OC(F)(F)F)cc3)c2cc1OC

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AXL P30530 18/20 0.58
EGFR P00533 1/20 0.55
MET P08581 1/20 0.55
SRC P12931 1/20 0.55
ALPL P05186 1/20 0.49
GSK3B P49841 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10328516 0.90 AXL (0.57) AXLEGFRMETSRCALPL
SCHEMBL13667478 0.89 AXL (0.57) AXLEGFRMETSRCALPL
SCHEMBL1592214 0.84 AXL (0.78) AXLEGFRMETSRC
SCHEMBL1590945 0.82 AXL (0.78) AXLEGFRMETSRC
SCHEMBL1591652 0.80 AXL (0.79) AXLEGFRMETSRC
SCHEMBL1591743 0.80 AXL (0.79) AXLEGFRMETSRC
SCHEMBL13667283 0.79 AXL (0.48) AXLEGFRMETSRC
SCHEMBL10328488 0.78 WDR5 (0.53) AXL
SCHEMBL13667556 0.78 AXL (0.70) AXLEGFRMETSRC
SCHEMBL10328505 0.77 AXL (0.73) AXLEGFRMETSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed
WO-2009127417-A1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2009-10-22 WO disclosed