SCHEMBL10334331

SCHEMBL10334331

CC1(C(=O)CBr)COc2cc(Cl)c(Cl)cc2O1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.37
ALPL P05186 2/20 0.34
CYP1A2 P05177 3/20 0.34
CYP2C19 P33261 3/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
MAPK1 P28482 1/20 0.33
NPC1 O15118 6/20 0.32
RAB9A P51151 6/20 0.32
SMN1; SMN2 Q16637 5/20 0.32
CHRM2 P08172 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
HPGD P15428 1/20 0.30
PPARA Q07869 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10334530 0.85 ALPG (0.38) NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL10334534 0.84 GPX4 (0.36) CYP3A4MAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL10334288 0.81 AKR1B1 (0.40) AKR1B1ALPLCYP1A2CYP2C19MAPK1
SCHEMBL10334289 0.81 AKR1B1 (0.38) AKR1B1ALPLCYP1A2CYP2C19CYP3A4
SCHEMBL10335039 0.79 ALOX15 (0.41) CYP1A2CYP2D6CYP2C9NPC1RAB9A
SCHEMBL10334527 0.78 HTR2B (0.41) CYP3A4MAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL10334538 0.67 KDM4E (0.38) CYP3A4MAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL10334332 0.67 ALOX15 (0.41) NPC1RAB9ASMN1; SMN2CHRM2CHRM1
SCHEMBL10334237 0.66 NPC1 (0.39) NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL10334301 0.66 NPC1 (0.39) NPC1RAB9ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4948797-A 2,2-disubstitued 2,3-dihydro-1,4-benzodioxin derivatives having hypotensive activity ISTITUTO LUSO FARMACO D'ITALIA S.P.A. (IT) 1990-08-14 US disclosed
EP-0367888-A1 2,2-Disubstituted 2,3-dihydro-1,4-benzodioxin derivatives having hypotensive activity ISTITUTO LUSO FARMACO D'ITALIA S.p.A. (IT) 1990-05-16 EP disclosed