SCHEMBL10334608

SCHEMBL10334608

CS(=O)(=O)Nc1cc2occ(NC=O)c(=O)c2cc1Oc1ccccc1F

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.76
ADORA3 P0DMS8 2/20 0.76
MIF P14174 1/20 0.76
PDE4A P27815 1/20 0.76
PDE4D Q08499 1/20 0.76
KMT2A Q03164 5/20 0.41
MEN1 O00255 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
PTGS2 P35354 3/20 0.40
CXCL8 P10145 1/20 0.36
CCR2 P41597 1/20 0.34
ALDH1A1 P00352 3/20 0.34
POLB P06746 1/20 0.34
KDM4E B2RXH2 3/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
ALDH2 P05091 1/20 0.33
RAB9A P51151 2/20 0.32
MAPT P10636 2/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10415468 0.89 ADORA3 (0.78) PTGS1ADORA3MIFPDE4APDE4D
Iguratimod SCHEMBL26326 0.87 PTGS1 (1.00) PTGS1ADORA3MIFPDE4APDE4D
Iguratimod SCHEMBL29366981 0.87 PTGS1 (1.00) PTGS1ADORA3MIFPDE4APDE4D
Iguratimod SCHEMBL5455197 0.86 PTGS1 (0.98) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL10416570 0.84 ADORA3 (0.54) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL7859528 0.83 ADORA3 (0.63) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL10415415 0.82 ADORA3 (0.52) PTGS1ADORA3MIFPDE4APDE4D
Iguratimod SCHEMBL29230458 0.81 PTGS1 (0.87) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL10417305 0.79 PTGS1 (0.85) PTGS1ADORA3MIFPDE4APDE4D
SCHEMBL30842776 0.78 PTGS1 (0.70) PTGS1ADORA3MIFPDE4APDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4954518-A Antiinflammatory agents TOYAMA CHEMICAL COMPANY, LTD. (JP) 1990-09-04 US claimed
JP-2049778-A None JP disclosed
JP-H0249778-A NOVEL 4H-1-BENZOPYRAN-4-ONE DERIVATIVE, ITS SALT AND ANTI-INFLAMMATORY AGENT CONTAINING THE SAME TOYAMA CHEM CO LTD 1990-02-20 JP disclosed