SCHEMBL7859528

SCHEMBL7859528

CS(=O)(=O)Nc1cc2occ(NC=O)c(=O)c2cc1Nc1ccccc1F

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.63
MIF P14174 1/20 0.63
PTGS1 P23219 1/20 0.63
PDE4A P27815 1/20 0.63
PDE4D Q08499 1/20 0.63
PLA2G7 Q13093 7/20 0.38
PTGS2 P35354 2/20 0.36
CDC25B P30305 1/20 0.34
ALDH2 P05091 1/20 0.33
BRD4 O60885 1/20 0.33
PSIP1 O75475 1/20 0.32
KEAP1 Q14145 1/20 0.32
FYN P06241 1/20 0.32
PKM P14618 1/20 0.31
ALDH1A1 P00352 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7859537 0.89 PTGS1 (0.56) ADORA3MIFPTGS1PDE4APDE4D
SCHEMBL10334608 0.83 PTGS1 (0.76) ADORA3MIFPTGS1PDE4APDE4D
SCHEMBL30842776 0.79 PTGS1 (0.70) ADORA3MIFPTGS1PDE4APDE4D
SCHEMBL29377983 0.78 ADORA3 (0.69) ADORA3MIFPTGS1PDE4APDE4D
SCHEMBL29377471 0.78 ADORA3 (0.69) ADORA3MIFPTGS1PDE4APDE4D
Iguratimod SCHEMBL26326 0.77 PTGS1 (1.00) ADORA3MIFPTGS1PDE4APDE4D
Potassium SCHEMBL29375000 0.77 ADORA3 (0.68) ADORA3MIFPTGS1PDE4APDE4D
Iguratimod SCHEMBL29366981 0.77 PTGS1 (1.00) ADORA3MIFPTGS1PDE4APDE4D
Iguratimod SCHEMBL5455197 0.76 PTGS1 (0.98) ADORA3MIFPTGS1PDE4APDE4D
SCHEMBL10415468 0.76 ADORA3 (0.78) ADORA3MIFPTGS1PDE4APDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0695547-B1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO LTD (JP) 2001-08-08 EP claimed
US-6166068-A Immunomodulator, cell adhesion inhibitor, and agent for treating, and preventing autoimmune diseases TOYAMA CHEMICAL CO., LTD. (JP) 2000-12-26 US claimed
US-5922755-A ADMINSTERING 4H-1-BENZOPYRAN-4-ONE DERIVATIVE TOYAMA CHEMICAL CO., LTD. (JP) 1999-07-13 US claimed
EP-0695547-A1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO., LTD. (JP) 1996-02-07 EP claimed
EP-0695547-B1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO LTD (JP) 2001-08-08 EP disclosed
US-6166068-A Immunomodulator, cell adhesion inhibitor, and agent for treating, and preventing autoimmune diseases TOYAMA CHEMICAL CO., LTD. (JP) 2000-12-26 US disclosed
US-5922755-A ADMINSTERING 4H-1-BENZOPYRAN-4-ONE DERIVATIVE TOYAMA CHEMICAL CO., LTD. (JP) 1999-07-13 US disclosed
EP-0695547-A1 IMMUNOMODULATOR, CELL ADHESION INHIBITOR, AND AGENT FOR TREATING AND PREVENTING AUTOIMMUNE DISEASES TOYAMA CHEMICAL CO., LTD. (JP) 1996-02-07 EP disclosed