SCHEMBL10340622

SCHEMBL10340622

N#Cc1cc(C(=O)O)n[nH]1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 15/20 0.52
DAO P14920 1/20 0.52
HCAR3 P49019 3/20 0.47
CYTH3 O43739 1/20 0.47
BTK Q06187 1/20 0.47
EPN1 Q9Y6I3 1/20 0.47
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24758142 0.82 HCAR2 (0.37) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL24117299 0.74 MAPK1 (0.39) HCAR2HCAR3MEN1KMT2APOLB
Water SCHEMBL1267709 0.72 HCAR2 (0.57) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL165390 0.72
Ammonia Solution, Strong SCHEMBL28463590 0.71 HCAR2 (0.55) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL165389 0.70
SCHEMBL70577 0.70 HCAR2 (0.59) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL220072 0.68
SCHEMBL19987833 0.68 HCAR2 (0.57) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL20929044 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250388601-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2025-12-25 US disclosed
US-12358928-B2 Compounds, compositions and methods DENALI THERAPEUTICS INC. (US) 2025-07-15 US disclosed
CN-118994191-A Inhibitors of receptor interacting protein kinase 1 戴纳立制药公司 2024-11-22 CN disclosed
CN-118994190-A Inhibitors of receptor interacting protein kinase 1 戴纳立制药公司 2024-11-22 CN disclosed
CN-114437105-B Inhibitors of receptor interacting protein kinase 1 戴纳立制药公司 2024-10-11 CN disclosed
US-20240150376-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2024-05-09 US disclosed
US-20230043400-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2023-02-09 US disclosed
US-20230043400-A1 Compounds, Compositions and Methods DENALI THERAPEUTICS INC. (US) 2023-02-09 US disclosed
CN-114437105-A Inhibitors of receptor interacting protein kinase 1 戴纳立制药公司 2022-05-06 CN disclosed
CN-109071504-B Inhibitors of receptor interacting protein kinase 1 戴纳立制药公司 2022-03-08 CN disclosed
WO-2017136727-A2 COMPOUNDS, COMPOSITIONS AND METHODS DENALI THERAPEUTICS INC. (US) 2017-08-10 WO disclosed
CN-1016398-B The pollen that contains pyrazole derivatives generates composite inhibiting ELLI LILLY & CO (US) 1992-04-29 CN disclosed
US-4966623-A POLLEN INHIBITION ACKMANN STEPHEN A (US) 1990-10-30 US disclosed
US-4902808-A HYBRID, POLLEN FORMATION INHIBITOR ELI LILLY AND COMPANY (US) 1990-02-20 US disclosed
EP-0177242-B1 POLLEN FORMATION INHIBITING PYRAZOLES ELI LILLY AND COMPANY (US) 1990-01-03 EP disclosed
US-4801326-A PRODUCTION OF HYBRID SEED ELI LILLY AND COMPANY (US) 1989-01-31 US disclosed
US-4775409-A PREVENTING POLLEN FORMATION ELI LILLY AND COMPANY (US) 1988-10-04 US disclosed
EP-0244075-A1 Gametocidal pyrazoles ELI LILLY AND COMPANY (US) 1987-11-04 EP disclosed
US-4666504-A HYBRIDS ELI LILLY AND COMPANY (US) 1987-05-19 US disclosed
EP-0177242-A2 Pollen formation inhibiting pyrazoles ELI LILLY AND COMPANY (US) 1986-04-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250388601-A1 Compounds, Compositions and Methods AURKC, WEE2, ERBB2 HCAR2 924/4885DAO 1600/4885HCAR3 1171/4885
US-20240150376-A1 Compounds, Compositions and Methods PIK3CA, PLK1, PIK3CB HCAR2 3504/4885DAO 4017/4885HCAR3 2641/4885
US-12358928-B2 Compounds, compositions and methods PIK3CA, PLK1, PIK3CB HCAR2 3504/4885DAO 4017/4885HCAR3 2641/4885
US-20230043400-A1 Compounds, Compositions and Methods PIK3CA, PLK1, PIK3CB HCAR2 3504/4885DAO 4017/4885HCAR3 2641/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.