SCHEMBL10344975

SCHEMBL10344975

CCc1cc(-c2n[nH]c(=S)n2-c2cccc3[nH]cnc23)c(O)cc1O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
HPGD P15428 3/20 0.43
LMNA P02545 1/20 0.43
ATM Q13315 1/20 0.43
HSP90AA1 P07900 9/20 0.42
HSP90AB1 P08238 2/20 0.42
KDM4E B2RXH2 2/20 0.39
MAPT P10636 2/20 0.39
GLA P06280 1/20 0.39
KMT2A Q03164 1/20 0.36
GAA P10253 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GFER P55789 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13983090 0.94 ALDH1A1 (0.41) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL12180265 0.83 HSP90AA1 (0.44) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL419118 0.82 ALDH1A1 (0.41) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL15042880 0.81 ALDH1A1 (0.40) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL14293304 0.80 HSP90AA1 (0.49) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL8931075 0.80 HSP90AA1 (0.49) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL8930611 0.79 HSP90AA1 (0.61) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL14344623 0.79 HSP90AA1 (0.48) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL12637703 0.79 HSP90AA1 (0.40) ALDH1A1HPGDLMNAATMHSP90AA1
SCHEMBL13983147 0.77 HSP90AA1 (0.43) ALDH1A1HPGDLMNAATMHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096919-A1 COMBINATION THERAPY OF HSP90 INHIBITORY COMPOUNDS WITH PROTEASOME INHIBITORS SYNTA PHARMACEUTICALS CORP. (US) 2012-07-19 WO disclosed
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO disclosed
WO-2011133520-A1 CANCER THERAPY USING A COMBINATION OF A HSP90 INHIBITORY COMPOUNDS AND A EGFR INHIBITOR SYNTA PHARMACEUTICALS CORP. (US) 2011-10-27 WO disclosed