SCHEMBL10345265

SCHEMBL10345265

CC(C)c1nc(-c2ccccc2)ccc1CO

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GCGR P47871 2/20 0.48
TRPV3 Q8NET8 1/20 0.40
NOTUM Q6P988 2/20 0.40
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ADORA1 P30542 4/20 0.39
PDCD1 Q15116 2/20 0.39
CD274 Q9NZQ7 2/20 0.39
ADORA3 P0DMS8 2/20 0.37
ADORA2A P29274 2/20 0.37
ADORA2B P29275 1/20 0.37
MAPT P10636 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
NPC1 O15118 1/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10589474 0.84 GCGR (0.50) GCGRTRPV3RAB9ANPC1SMN1; SMN2
SCHEMBL14943937 0.77 ALDH1A1 (0.54) NOTUMRAB9AMEN1KMT2AALDH1A1
SCHEMBL14931897 0.76 PDCD1 (0.41) TRPV3RAB9AMEN1KMT2AALDH1A1
SCHEMBL20885480 0.74 MEN1 (0.43) GCGRRAB9AMEN1KMT2AALDH1A1
SCHEMBL3210688 0.74 MEN1 (0.43) NOTUMRAB9AMEN1KMT2AALDH1A1
SCHEMBL12427062 0.73 SQOR (0.53) RAB9AMEN1KMT2AALDH1A1PDCD1
SCHEMBL12413897 0.72 GCGR (0.35) GCGRALDH1A1CD274
SCHEMBL12427066 0.71 HSD17B10 (0.50) RAB9AMEN1KMT2AALDH1A1PDCD1
SCHEMBL10345761 0.71 HPGD (0.49) GCGRALDH1A1ADORA1ADORA2A
SCHEMBL12427064 0.71 SQOR (0.52) NOTUMRAB9AMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0356788-A2 Quinoline and pyridine anchors for HMG-CoA reductase inhibitors E.R. SQUIBB & SONS, INC. (US) 1990-03-07 EP disclosed