SCHEMBL10349779

SCHEMBL10349779

C=CN(CC(=O)OC)C(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.48
ALDH1A1 P00352 5/20 0.45
MAPK1 P28482 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TGM2 P21980 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CCR6 P51684 1/20 0.41
PAX8 Q06710 1/20 0.41
F13A1 P00488 1/20 0.41
TGM1 P22735 1/20 0.41
LMNA P02545 2/20 0.41
HCAR2 Q8TDS4 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KMT2A Q03164 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236855 0.85 ALDH1A1 (0.46) ALDH1A1MAPK1L3MBTL1TGM2CCR6
SCHEMBL10494016 0.85 HCAR2 (0.47) ALDH1A1HCAR2KMT2AKDM4E
SCHEMBL10382170 0.81 ABCB1 (0.46) ABCB1ALDH1A1MAPK1L3MBTL1TGM2
SCHEMBL8473781 0.80 L3MBTL1 (0.46) ALDH1A1MAPK1L3MBTL1SMN1; SMN2LMNA
SCHEMBL13675129 0.80 ALDH1A1 (0.47) ALDH1A1MAPK1L3MBTL1TGM2SMN1; SMN2
SCHEMBL16207467 0.80 ABCB1 (0.50) ABCB1ALDH1A1MAPK1L3MBTL1SMN1; SMN2
SCHEMBL25461074 0.80 ABCB1 (0.55) ABCB1ALDH1A1MAPK1L3MBTL1TGM2
SCHEMBL5069687 0.77 ALDH1A1 (0.50) ABCB1ALDH1A1MAPK1L3MBTL1SMN1; SMN2
SCHEMBL19189188 0.77 CCR6 (0.49) ABCB1ALDH1A1MAPK1L3MBTL1CCR6
SCHEMBL13603924 0.75 ALDH1A1 (0.51) ABCB1ALDH1A1MAPK1L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0238245-B1 3-HALOVINYLGLYCINE ANTIBACTERIAL AGENTS MERCK & CO. INC. (US) 1990-06-20 EP disclosed
US-4806680-A REACTING IN N-PROTECTED VINYLGLYCINE ESTER WITH ARYLSELENENYL HALIDE, OXIDATION THE ADDUCT, HEATING IN MINERAL ACID MERCK & CO., INC. (US) 1989-02-21 US disclosed
US-4727062-A INHIBITORS OF ALANINE RACEMASE MERCK & CO., INC. (US) 1988-02-23 US disclosed
EP-0238245-A1 3-Halovinylglycine antibacterial agents MERCK & CO. INC. (US) 1987-09-23 EP disclosed