SCHEMBL10355347

SCHEMBL10355347

COc1cccc(-c2nc(CO)c[nH]2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DCUN1D1 Q96GG9 1/20 0.49
PIN1 Q13526 1/20 0.48
GRK6 P43250 1/20 0.46
AURKA O14965 1/20 0.46
NR1H2 P55055 1/20 0.46
NR1H3 Q13133 1/20 0.46
NR1I2 O75469 1/20 0.45
CYP1A2 P05177 1/20 0.45
VDR P11473 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2B6 P20813 1/20 0.45
AHR P35869 1/20 0.45
NR1I3 Q14994 1/20 0.45
PARP1 P09874 1/20 0.44
DYRK1A Q13627 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
NTRK1 P04629 1/20 0.43
TYMP P19971 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28289637 0.81 PDGFRB (0.54) DCUN1D1PIN1AURKANR1H2NR1H3
SCHEMBL10556612 0.81 KDM4E (0.46) AURKAMAPTSMN1; SMN2KDM4ETDP1
SCHEMBL20425457 0.80 DCUN1D1 (0.52) DCUN1D1PIN1AURKANR1H2NR1H3
SCHEMBL10099697 0.77 PDGFRB (0.50) DCUN1D1GRK6DYRK1ACLK4ADORA2A
SCHEMBL7192429 0.77 KIF11 (0.44) PIN1DYRK1A
SCHEMBL7254835 0.77 IDO1 (0.46) DYRK1A
SCHEMBL2549690 0.76 GRK6 (0.48) GRK6DYRK1A
SCHEMBL7146244 0.76 NR1H2 (0.58) DCUN1D1PIN1NR1H2NR1H3NR1I2
SCHEMBL672597 0.76 NOTUM (0.42) DCUN1D1PIN1NR1H2NR1H3CYP1A2
SCHEMBL15332174 0.75 ALDH1A1 (0.56) DCUN1D1PIN1AURKANR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0074130-B1 NEW IMIDAZOLE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ZAMBON S.p.A. (IT) 1990-09-19 EP disclosed