SCHEMBL10356189

SCHEMBL10356189

CC[C@]12CC[C@@H]3c4ccc(OC)cc4CC[C@H]3[C@@H]1C=CC2=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.56
HSD17B1 P14061 2/20 0.56
MAPT P10636 2/20 0.56
RECQL P46063 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
HSD17B10 Q99714 1/20 0.50
ESR1 P03372 4/20 0.48
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
HIF1A Q16665 1/20 0.47
NR3C1 P04150 1/20 0.47
PGR P06401 1/20 0.47
CNR1 P21554 1/20 0.47
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
SLC6A3 Q01959 1/20 0.47
ALDH1A1 P00352 2/20 0.45
PDE4D Q08499 1/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2360694 0.86 ESR1 (0.54) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL2738485 0.84 LMNA (0.67) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL12164090 0.84 LMNA (0.67) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL5024803 0.84 LMNA (0.67) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL6570384 0.83 LMNA (0.40) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL6570381 0.83 LMNA (0.40) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL11862021 0.82 LMNA (0.72) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL11857394 0.82 LMNA (0.72) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL11857389 0.82 LMNA (0.72) LMNAHSD17B1MAPTRECQLSMN1; SMN2
SCHEMBL4623091 0.82 LMNA (0.72) LMNAHSD17B1MAPTRECQLSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0285548-B1 PROCESS FOR THE PREPARATION OF 17-ALPHA-ETHYNYL-17-BETA-HYDROXY-18-METHYL-4,15-ESTRADIEN-3-ONE, AND INTERMEDIATES FOR THIS PROCESS SCHERING AKTIENGESELLSCHAFT (DE) 1990-09-05 EP claimed
EP-0285548-A1 Process for the preparation of 17-alpha-ethynyl-17-beta-hydroxy-18-methyl-4,15-estradien-3-one, and intermediates for this process SCHERING AKTIENGESELLSCHAFT (DE) 1988-10-05 EP claimed
EP-0285548-B1 PROCESS FOR THE PREPARATION OF 17-ALPHA-ETHYNYL-17-BETA-HYDROXY-18-METHYL-4,15-ESTRADIEN-3-ONE, AND INTERMEDIATES FOR THIS PROCESS SCHERING AKTIENGESELLSCHAFT (DE) 1990-09-05 EP disclosed
US-4923640-A Process for the production of 17α-ethinyl-17β-hydroxy-18-methyl-4,15-estradien-3-one and new intermediate products for this process SCHERING AKTIENGESELLSCHAFT (DE) 1990-05-08 US disclosed
EP-0285548-A1 Process for the preparation of 17-alpha-ethynyl-17-beta-hydroxy-18-methyl-4,15-estradien-3-one, and intermediates for this process SCHERING AKTIENGESELLSCHAFT (DE) 1988-10-05 EP disclosed