SCHEMBL10356744

SCHEMBL10356744

CCN(CC)CCOc1ccc(C(O)(CC)c2ccccc2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.58
HTT P42858 2/20 0.58
CYP1A2 P05177 2/20 0.58
CYP2C9 P11712 2/20 0.58
LTA4H P09960 1/20 0.58
CYP2C19 P33261 1/20 0.58
SIGMAR1 Q99720 5/20 0.56
EBP Q15125 4/20 0.56
KMT2A Q03164 4/20 0.54
CHRM2 P08172 4/20 0.54
CHRM1 P11229 4/20 0.54
ESR1 P03372 4/20 0.54
MEN1 O00255 3/20 0.54
CHRM3 P20309 3/20 0.54
KDM4E B2RXH2 3/20 0.54
KCNH2 Q12809 2/20 0.54
ADRA2A P08913 2/20 0.54
ADORA3 P0DMS8 2/20 0.54
PTGS1 P23219 2/20 0.54
SLC6A2 P23975 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tribromoethanol SCHEMBL11621823 0.94 CYP2D6 (0.52) CYP2D6HTTCYP1A2CYP2C9LTA4H
Fumaric Acid SCHEMBL11622225 0.91 BCHE (0.55) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL16910242 0.88 SIGMAR1 (0.69) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL10878286 0.87 EBP (0.72) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL10880656 0.87 EBP (0.55) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL10877202 0.86 EBP (0.49) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL10878610 0.86 EBP (0.57) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL10879788 0.84 KMT2A (0.53) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL10893666 0.84 EBP (0.52) CYP2D6HTTCYP1A2CYP2C9LTA4H
SCHEMBL330094 0.83 SIGMAR1 (0.67) CYP2D6HTTCYP1A2CYP2C9LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0112587-B1 DERIVATIVES OF 4-(1-(PHENYL)-1-(HYDROXY)-PROP-1-YL)-RESORCINE, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THESE COMPOUNDS RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 1990-09-19 EP disclosed
EP-0112588-B1 4-HYDROXY-ALPHA-ETHYL BENZHYDROLES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THESE COMPOUNDS RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 1987-11-11 EP disclosed
US-4094908-A Alpha-substituted benzhydrol derivatives RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1978-06-13 US disclosed
US-4039589-A LIVER MICROSOMAL ENZYMES RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1977-08-02 US disclosed