SCHEMBL10358301

SCHEMBL10358301

Cc1ccc2sc(C3CC(=O)NC3=S)nc2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.39
SIRT1 Q96EB6 1/20 0.38
MAPT P10636 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36
IDO1 P14902 2/20 0.36
LMNA P02545 3/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
PKM P14618 1/20 0.36
CCR6 P51684 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 3/20 0.33
ROCK2 O75116 1/20 0.33
GAA P10253 2/20 0.33
ALOX12 P18054 1/20 0.32
UBE2M P61081 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10358336 0.78 SMN1; SMN2 (0.41) MAPTSMN1; SMN2TP53LMNANPC1
SCHEMBL10759361 0.78 DYRK1A (0.39) DYRK1AMAPTSMN1; SMN2TP53LMNA
SCHEMBL10358298 0.69 DDB1 (0.41) DYRK1AMAPTSMN1; SMN2TP53IDO1
SCHEMBL20135675 0.68 NPC1 (0.68) DYRK1AMAPTSMN1; SMN2TP53LMNA
SCHEMBL29688848 0.68 NPC1 (0.68) DYRK1AMAPTSMN1; SMN2TP53LMNA
SCHEMBL26567985 0.67 MAPT (0.43) DYRK1AMAPTSMN1; SMN2TP53LMNA
SCHEMBL13082023 0.67 NPC1 (0.49) DYRK1AMAPTSMN1; SMN2TP53LMNA
SCHEMBL23010591 0.64 UBE2M (0.50) MAPTSMN1; SMN2TP53LMNANPC1
SCHEMBL26049456 0.63 DDB1 (0.43)
SCHEMBL92781 0.63 SMN1; SMN2 (0.61) DYRK1AMAPTSMN1; SMN2TP53LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161222-B1 HETEROCYCLIC MERCAPTOCARBOXYLIC-ACID AMIDES, IMIDES AND NITRILES AS CORROSION INHIBITING AGENTS CIBA-GEIGY AG (CH) 1990-10-10 EP disclosed
US-4719036-A PAINTS; METAL WORKING CIBA-GEIGY CORPORATION (US) 1988-01-12 US disclosed
EP-0161222-A2 Heterocyclic mercaptocarboxylic-acid amides, imides and nitriles as corrosion inhibiting agents CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed