SCHEMBL10358705

SCHEMBL10358705

Fc1ccc(C(Br)c2ccc(C(F)(F)F)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.42
CYP19A1 P11511 1/20 0.42
PAX8 Q06710 1/20 0.41
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
PDE2A O00408 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
ACP3 P15309 1/20 0.38
TACR1 P25103 2/20 0.38
SLC6A9 P48067 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
KIF11 P52732 1/20 0.37
USP2 O75604 1/20 0.36
RAB9A P51151 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4428819 0.91 GSK3B (0.48) GSK3BCES2CES1PDE2AACP3
SCHEMBL4427290 0.83 IDO1 (0.46) CYP19A1CES2CES1ALDH1A1
SCHEMBL7523008 0.83 ACP3 (0.55) GSK3BACP3ALDH1A1TSHRKIF11
SCHEMBL168026 0.81 ALDH1A1 (0.53) PAX8CES2CES1CYP1A1CYP1B1
SCHEMBL23040160 0.79 CYP19A1 (0.38) CYP19A1PDE2ATSHR
Bromomethane SCHEMBL27825372 0.79 PAX8 (0.47) GSK3BPAX8CES2CES1CYP1A1
SCHEMBL23960462 0.78 PDE2A (0.47) CYP19A1PAX8CES2CES1PDE2A
SCHEMBL23960467 0.78 PDE2A (0.47) CYP19A1PAX8CES2CES1PDE2A
SCHEMBL1350356 0.78 PAX8 (0.49) CYP19A1PAX8CES2CES1PDE2A
SCHEMBL23960464 0.78 PDE2A (0.47) CYP19A1PAX8CES2CES1PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0243904-B1 Optionally substituted 1-(2'-[bis-(phenyl)-methoxy]-ethyl)-4-(3'[bis-(phenyl)-methoxy]propyl)piperazines, process for their preparation and medicines containing them Richter Gedeon Vegyészeti Gyár R.T. (HU) 1990-10-31 EP disclosed
US-4866062-A TREATMENT OF DISEASES ARISING FROM A HYPOFUNCTION OF THE DOPAMINERGIC SYSTEM RICHTER GEDEON VEGYESZETI GYAR (HU) 1989-09-12 US disclosed
EP-0243904-A1 Optionally substituted 1-(2'-[bis-(phenyl)-methoxy]-ethyl)-4-(3'[bis-(phenyl)-methoxy]propyl)piperazines, process for their preparation and medicines containing them Richter Gedeon Vegyészeti Gyár R.T. (HU) 1987-11-04 EP disclosed