SCHEMBL10360876

SCHEMBL10360876

CC/N=N/Nc1ccc(C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.43
NPC1 O15118 5/20 0.40
RAB9A P51151 5/20 0.40
ALDH1A1 P00352 5/20 0.40
GAA P10253 5/20 0.40
TDP1 Q9NUW8 4/20 0.40
HPGD P15428 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KYAT1 Q16773 1/20 0.39
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
GFER P55789 2/20 0.37
HTT P42858 2/20 0.37
DHODH Q02127 1/20 0.36
LMNA P02545 2/20 0.35
ACHE P22303 1/20 0.35
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1278598 1.00 MAPT (0.43) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL1278595 1.00 MAPT (0.43) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL10840042 0.83 MAPT (0.40) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL1278625 0.83 MAPT (0.40) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL1278627 0.83 MAPT (0.40) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL7343923 0.82 SCN5A (0.40) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL1887617 0.82 SCN5A (0.40) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL3501691 0.80 TSHR (0.50) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL7369814 0.76 TGM2 (0.38) MAPTNPC1RAB9AALDH1A1GAA
SCHEMBL7369817 0.76 TGM2 (0.38) MAPTNPC1RAB9AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0139614-B1 PHARMACEUTICAL PREPARATIONS CONTAINING FLAVANONE OR THIOFLAVANONE DERIVATIVES, THE USE THEREOF, NOVEL FLAVANONES AND THIOFLAVANONES, AND PROCESSES FOR THEIR MANUFACTURE Zyma SA (CH) 1990-08-22 EP disclosed
US-4885298-A Pharmaceutical preparations containing flavanone or thioflavanone derivatives the use thereof, novel flavanones and thioflavanones, and processes for their manufacture ZYMA SA (CH) 1989-12-05 US disclosed
EP-0096008-B1 (+)-CYANIDAN-3-OL DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE, PHARMACEUTICAL PREPARATIONS THAT CONTAIN SUCH COMPOUNDS, AND THE USE OF THE LATTER Zyma SA (CH) 1989-03-29 EP disclosed
US-4644011-A LIVER AND VIEN DISORDERS ZYMA SA (CH) 1987-02-17 US disclosed
US-4595677-A Substituted tetrapeptides CIBA-GEIGY CORPORATION (US) 1986-06-17 US disclosed
US-4579684-A Process for the manufacture of enol derivatives CIBA-GEIGY CORPORATION (US) 1986-04-01 US disclosed
US-4552871-A ALDOSTERONE-ANTAGONISTIC, DIURETICS CIBA GEIGY CORPORATION (US) 1985-11-12 US disclosed
US-4510159-A (+)-Cyanidan-3-ol derivatives, pharmaceutical preparations that contain such compounds, and the use of the latter to treat liver or venous diseases ZYMA SA (CH) 1985-04-09 US disclosed
EP-0115473-A2 Substituted pyrrolidinone derivatives and process for their preparation CIBA-GEIGY AG (CH) 1984-08-08 EP disclosed
EP-0115472-A2 Pyrrolidinon derivatives and process for their preparation CIBA-GEIGY AG (CH) 1984-08-08 EP disclosed
US-4405778-A Process for preparing cephalosporin ethers CIBA-GEIGY CORPORATION (US) 1983-09-20 US disclosed
US-4319027-A Process for the manufacture of ceohem enol derivatives CIBA-GEIGY CORPORATION (US) 1982-03-09 US disclosed
EP-0045281-A1 Triazoline derivatives and processes for their preparation CIBA-GEIGY AG (CH) 1982-02-03 EP disclosed
US-4313945-A 7-Thiazolyl-acetamido-cephem derivatives with terminal aminocarboxylic acid grouping CIBA-GEIGY CORPORATION (US) 1982-02-02 US disclosed
US-4301278-A BY HYDROGENATION IN THE PRESENCE OF A CATALYST CIBA-GEIGY CORPORATION (US) 1981-11-17 US disclosed
US-4293462-A Process for the manufacture of enol derivatives, and intermediates CIBA-GEIGY CORPORATION (US) 1981-10-06 US disclosed
US-4256739-A 7β-Amino-3-thio-3-cephem-4-carboxylic acid compounds, and antibacterial compositions and methods using them CIBA-GEIGY CORPORATION (US) 1981-03-17 US disclosed
US-4255328-A CEPHALOSPORINS CIBA-GEIGY CORPORATION (US) 1981-03-10 US disclosed
US-4110533-A PROCESS FOR THE MANUFACTURE OF ENOL DERIVATIVES CIBA-GEIGY CORPORATION (US) 1978-08-29 US disclosed
US-4073902-A ANTIMICROBIAL COMPOUNDS CIBA-GEIGY CORPORATION (US) 1978-02-14 US disclosed