SCHEMBL10364503

SCHEMBL10364503

COC(=O)c1ccc(Cl)cc1NC(=O)NC(C)C

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.57
KMT2A Q03164 5/20 0.54
MEN1 O00255 4/20 0.54
LMNA P02545 2/20 0.54
ALDH1A1 P00352 8/20 0.52
KDM4E B2RXH2 4/20 0.52
NPSR1 Q6W5P4 1/20 0.52
ABL1 P00519 1/20 0.51
HPGD P15428 3/20 0.50
TP53 P04637 2/20 0.49
HTT P42858 1/20 0.49
GRIK1 P39086 2/20 0.49
RAB9A P51151 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9227218 0.85 ALDH1A1 (0.71) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL10363345 0.84 KDM4E (0.54) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL27203069 0.84 KDM4E (0.74) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL10364417 0.84 KDM4E (0.54) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL9510448 0.83 GAA (0.53) MAPTKMT2ALMNAALDH1A1KDM4E
SCHEMBL10363762 0.82 KDM4E (0.53) MAPTKMT2ALMNAALDH1A1KDM4E
SCHEMBL10362862 0.81 SMN1; SMN2 (0.57) KMT2AMEN1LMNAALDH1A1KDM4E
SCHEMBL5928755 0.80 ABL1 (0.58) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL7256022 0.79 KCNMA1 (0.55) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL10362881 0.79 KDM4E (0.76) MAPTKMT2AMEN1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0147211-B1 4H-3,1-BENZOXAZIN-4-ONES AND RELATED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES FOR THEIR PREPARATION SYNTEX (U.S.A.) INC. (US) 1990-09-12 EP disclosed
US-4657893-A ANTIINFLAMMATORY AGENTS SYNTEX (U.S.A.) INC. (US) 1987-04-14 US disclosed
EP-0147211-A2 4H-3,1-benzoxazin-4-ones and related compounds, pharmaceutical compositions containing them, and processes for their preparation SYNTEX (U.S.A.) INC. (US) 1985-07-03 EP disclosed