SCHEMBL10364950

SCHEMBL10364950

CC1=C(C(=O)O)C(c2ccc([N+](=O)[O-])cc2)C(C(=O)OC2(C)CCCO2)=C(C)N1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.54
ADORA3 P0DMS8 2/20 0.52
ADRA1A P35348 8/20 0.45
ADRA2A P08913 7/20 0.45
ADRA2B P18089 7/20 0.45
ADRA2C P18825 7/20 0.45
ADRA1D P25100 7/20 0.45
ADRA1B P35368 7/20 0.45
CACNA1F O60840 2/20 0.44
CACNA1D Q01668 2/20 0.44
CACNA1S Q13698 2/20 0.44
CACNA1C Q13936 2/20 0.44
TDP1 Q9NUW8 1/20 0.43
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
NOTCH1 P46531 1/20 0.42
PSEN1 P49768 1/20 0.42
PSEN2 P49810 1/20 0.42
CCNA1 P78396 1/20 0.42
APH1B Q8WW43 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7416445 0.89 CACNA1F (0.58) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7424363 0.83 ADORA3 (0.58) CACNA1BADORA3ADRA1ACACNA1FCACNA1D
SCHEMBL10671428 0.81 MEN1 (0.65) ADORA3CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7034433 0.80 CACNA1B (0.64) CACNA1BADORA3ADRA1AADRA2AADRA2B
SCHEMBL7433908 0.80 CACNA1C (0.64) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL7160127 0.79 ADORA3 (0.78) CACNA1BADORA3ADRA1AADRA2AADRA2B
SCHEMBL7235504 0.78 CACNA1B (0.59) CACNA1BADORA3ADRA1AADRA2AADRA2B
SCHEMBL10669458 0.76 CACNA1C (0.59) CACNA1BADORA3CACNA1FCACNA1DCACNA1S
SCHEMBL10364949 0.76 KMT2A (0.65) CACNA1BADORA3MEN1ALDH1A1LMNA
SCHEMBL9673699 0.76 KDM4E (0.43) TDP1MEN1ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0126094-B1 NEW 1,4-DIHYDROPYRIDINE ESTERS AND PREPARATION METHODS THEREOF AND DRUGS CONTAINING SAID ESTERS CERMOL S.A. (CH) 1990-06-20 EP disclosed