SCHEMBL10367108

SCHEMBL10367108

Cc1cc(Br)cnc1NCCCCN

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
STK17A Q9UEE5 14/20 0.47
SYK P43405 3/20 0.43
AURKA O14965 1/20 0.40
JAK1 P23458 1/20 0.40
KDR P35968 1/20 0.40
KCNH2 Q12809 1/20 0.40
LRRK2 Q5S007 1/20 0.40
AURKB Q96GD4 1/20 0.40
STK17B O94768 5/20 0.39
BRD4 O60885 2/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10365100 0.95 STK17A (0.51) STK17ASYKSTK17BNPC1ALDH1A1
SCHEMBL10732356 0.81 STK17A (0.48) STK17ASYKAURKAJAK1KDR
SCHEMBL10365097 0.79 MAPT (0.47) STK17ASYKSTK17BNPC1ALDH1A1
SCHEMBL10732016 0.79 STK17A (0.47) STK17ASYKAURKAJAK1KDR
SCHEMBL10366902 0.78 STK17A (0.33) STK17ASYKNPC1ALDH1A1
SCHEMBL19260116 0.76 ALDH1A1 (0.40) NPC1ALDH1A1
SCHEMBL10367439 0.76 STK17A (0.51) STK17ASTK17B
SCHEMBL10731426 0.76 STK17A (0.51) STK17ASYKSTK17B
SCHEMBL10365885 0.76 STK17A (0.33) STK17ASYKNPC1ALDH1A1
SCHEMBL7751879 0.75 ALDH1A1 (0.40) STK17AAURKAKDRLRRK2AURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206623-B1 PYRIDINE DERIVATIVES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-10-24 EP disclosed
US-4771058-A ANTIHISTAMINES SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1988-09-13 US disclosed
EP-0206623-A2 Pyridine derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-12-30 EP disclosed