SCHEMBL10368285

SCHEMBL10368285

COC(=O)OC1=C(C)NC(C)=C([N+](=O)[O-])C1c1ccccc1OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.45
CYP1A2 P05177 5/20 0.45
CYP3A4 P08684 4/20 0.45
MAPT P10636 4/20 0.45
CYP2C9 P11712 4/20 0.45
CYP2C19 P33261 4/20 0.45
CACNA1C Q13936 4/20 0.45
TSHR P16473 3/20 0.45
NFKB1 P19838 3/20 0.45
CYP2D6 P10635 2/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ABCC4 O15439 2/20 0.41
CACNA1F O60840 2/20 0.41
ABCB11 O95342 2/20 0.41
LMNA P02545 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10914095 0.89 POLB (0.46) MAPTKMT2AMEN1KDM4ESMN1; SMN2
SCHEMBL10501976 0.87 PDE1C (0.38) ADORA3CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL10502844 0.87 PDE1C (0.38) ADORA3CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL10351329 0.86 CYP1A2 (0.41) ADORA3CYP1A2CYP3A4MAPTCYP2C9
Alcohol SCHEMBL9690926 0.86 MAPT (0.48) ADORA3CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL9690807 0.86 POLB (0.44) MAPTKMT2AMEN1KDM4ESMN1; SMN2
SCHEMBL9691359 0.86 POLB (0.44) MAPTKMT2AMEN1KDM4ESMN1; SMN2
SCHEMBL11023305 0.86 MTNR1A (0.40) ADORA3CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL10647063 0.85 POLB (0.43) MAPTKMT2AMEN1KDM4ESMN1; SMN2
SCHEMBL9690786 0.84 MEN1 (0.48) ADORA3CYP1A2CYP3A4MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0186028-B1 OPTICALLY ACTIVE NITRODIHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN MEDICINES BAYER AG (DE) 1990-08-01 EP disclosed
EP-0186028-A2 Optically active nitrodihydropyridines, process for their preparation and their use in medicines BAYER AG (DE) 1986-07-02 EP disclosed