SCHEMBL10501976

SCHEMBL10501976

CC1=C(OC(=O)OCCCCCCN)C(c2ccccc2OCc2ccccc2)C([N+](=O)[O-])=C(C)N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 1/20 0.38
CACNA1C Q13936 8/20 0.37
ADORA3 P0DMS8 4/20 0.37
CYP1A2 P05177 3/20 0.37
CYP3A4 P08684 3/20 0.37
MAPT P10636 3/20 0.37
CYP2C9 P11712 3/20 0.37
CYP2C19 P33261 3/20 0.37
KMT2A Q03164 3/20 0.37
TSHR P16473 2/20 0.37
NFKB1 P19838 2/20 0.37
MEN1 O00255 2/20 0.37
CYP2D6 P10635 1/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CACNA1F O60840 6/20 0.36
CACNA1D Q01668 6/20 0.36
CACNA1S Q13698 6/20 0.36
SIRT1 Q96EB6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10502844 1.00 PDE1C (0.38) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL11023305 0.90 MTNR1A (0.40) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL10734668 0.88 PDE1C (0.47) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL10730896 0.88 PDE1C (0.47) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL10368285 0.87 ADORA3 (0.45) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL10868953 0.84 TP53 (0.38) CACNA1CKMT2ATSHRMEN1TP53
SCHEMBL10517437 0.82 NR1I2 (0.43) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL10351329 0.81 CYP1A2 (0.41) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL10516700 0.81 NR1I2 (0.44) PDE1CCACNA1CADORA3CYP1A2CYP3A4
SCHEMBL10734312 0.81 PDE1C (0.50) PDE1CCACNA1CADORA3CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0164010-B1 3-NITRO-DIHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION AND THEIR PHARMACEUTICAL USE BAYER AG (DE) 1989-02-22 EP disclosed
EP-0164010-A2 3-Nitro-dihydropyridines, process for their preparation and their pharmaceutical use BAYER AG (DE) 1985-12-11 EP disclosed