SCHEMBL10370210

SCHEMBL10370210

O=C(CCCN1CC2C3C=CC(C4CC34)C2C1)c1ccc(F)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 3/20 0.56
HTR1A P08908 2/20 0.56
MEN1 O00255 1/20 0.56
CHRM2 P08172 1/20 0.56
ADRA2A P08913 1/20 0.56
DRD1 P21728 1/20 0.56
ADRA1A P35348 1/20 0.56
OPRM1 P35372 1/20 0.56
KMT2A Q03164 1/20 0.56
KCNH2 Q12809 1/20 0.56
HRH3 Q9Y5N1 1/20 0.56
DRD2 P14416 6/20 0.56
DRD4 P21917 1/20 0.56
TSHR P16473 1/20 0.55
KDM4E B2RXH2 1/20 0.54
HSD17B10 Q99714 1/20 0.54
NPC1 O15118 1/20 0.54
RAB9A P51151 1/20 0.54
HTR2A P28223 2/20 0.51
CYP2D6 P10635 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10372093 0.92 DRD3 (0.60) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL10370891 0.92 DRD3 (0.59) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL10397519 0.81 DRD3 (0.58) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL4501475 0.80 DRD3 (0.71) DRD3HTR1AMEN1CHRM2ADRA2A
Nonaperone SCHEMBL2109345 0.80 DRD3 (0.67) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL8989763 0.79 DRD3 (0.53) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL8989690 0.79 DRD2 (0.67) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL7781094 0.76 DRD2 (0.60) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL4496558 0.75 TSHR (0.76) DRD3HTR1AMEN1CHRM2ADRA2A
SCHEMBL8989694 0.75 DRD2 (0.53) DRD3DRD2DRD4KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4937347-A Polycyclicamine with psychotropic activity AMERICAN HOME PRODUCTS CORPORATION (US) 1990-06-26 US disclosed
US-4927934-A Polycyclicamine with psychotropic activity AMERICAN HOME PRODUCTS CORPORATION (US) 1990-05-22 US disclosed
EP-0348460-A1 POLYCYCLICAMINES WITH PSYCHOTROPIC ACTIVITY AMERICAN HOME PRODUCTS CORPORATION (US) 1990-01-03 EP disclosed
US-4855430-A Polycyclicamine with psychotropic activity AMERICAN HOME PRODUCTS CORPORATION (US) 1989-08-08 US disclosed