SCHEMBL10372811

SCHEMBL10372811

CSc1sc2ccccc2c1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.44
MAPT P10636 5/20 0.37
RAB9A P51151 5/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
KDM4E B2RXH2 4/20 0.37
NPC1 O15118 3/20 0.37
PTGS2 P35354 2/20 0.37
ALDH1A1 P00352 3/20 0.36
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
MAOB P27338 2/20 0.33
NFKB1 P19838 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
HPGD P15428 1/20 0.33
MAOA P21397 1/20 0.33
LMNA P02545 2/20 0.33
PTPN1 P18031 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9266269 0.78 GPR3 (0.46) GPR3MAPTRAB9AMEN1KMT2A
SCHEMBL718497 0.72 GPR3 (0.50) GPR3MAPTRAB9AMEN1KMT2A
SCHEMBL10375309 0.72 GPR3 (0.40) GPR3KDM4ENPC1ALDH1A1TDP1
SCHEMBL29434786 0.72 GPR3 (0.55) GPR3MAPTRAB9AMEN1KMT2A
SCHEMBL1518983 0.72 GPR3 (0.55) GPR3MAPTRAB9AMEN1KMT2A
SCHEMBL309376 0.72 GPR3 (0.55) GPR3MAPTRAB9AMEN1KMT2A
SCHEMBL3123867 0.71 LIMK1 (0.38) RAB9AMEN1KMT2AKDM4ENPC1
SCHEMBL19135547 0.70 GPR3 (0.52) GPR3MAPTRAB9AMEN1KMT2A
SCHEMBL9272736 0.68 EGFR (0.43) GPR3MAPTRAB9AMEN1KMT2A
SCHEMBL24442088 0.68 GPR3 (0.50) GPR3MAPTRAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0217530-B1 DIHYDROPYRIDINES ELI LILLY AND COMPANY (US) 1990-10-31 EP disclosed
US-4659717-A CAUSING VASODILATION ELI LILLY AND COMPANY (US) 1987-04-21 US disclosed
EP-0217530-A1 Dihydropyridines ELI LILLY AND COMPANY (US) 1987-04-08 EP disclosed